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TRPV1 channels are intrinsically heat sensitive and negatively regulated by phosphoinositide lipids

The capsaicin receptor, TRPV1, is regulated by phosphatidylinositol-4,5-bisphosphate (PIP(2)), although the precise nature of this effect (i.e., positive or negative) remains controversial. Here, we reconstitute purified TRPV1 into artificial liposomes, where it is gated robustly by capsaicin, proto...

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Bibliografski detalji
Glavni autori: Cao, Erhu, Cordero-Morales, Julio F., Liu, Beiying, Qin, Feng, Julius, David
Format: Artigo
Jezik:Inglês
Izdano: 2013
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3583019/
https://ncbi.nlm.nih.gov/pubmed/23439120
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuron.2012.12.016
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