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Explaining why Gleevec is a specific and potent inhibitor of Abl kinase

Tyrosine kinases present attractive drug targets for specific types of cancers. Gleevec, a well-known therapeutic agent against chronic myelogenous leukemia, is an effective inhibitor of Abl tyrosine kinase. However, Gleevec fails to inhibit closely homologous tyrosine kinases, such as c-Src. Becaus...

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Autors principals: Lin, Yen-Lin, Meng, Yilin, Jiang, Wei, Roux, Benoît
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3562763/
https://ncbi.nlm.nih.gov/pubmed/23319661
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1214330110
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