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Molecular sampling of the allosteric binding pocket of the TSH receptor provides discriminative pharmacophores for antagonist and agonists

The TSHR (thyrotropin receptor) is activated endogenously by the large hormone thyrotropin and activated pathologically by auto-antibodies. Both activate and bind at the extracellular domain. Recently, SMLs (small-molecule ligands) have been identified, which bind in an allosteric binding pocket wit...

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Detalhes bibliográficos
Main Authors: Hoyer, Inna, Haas, Ann-Karin, Kreuchwig, Annika, Schülein, Ralf, Krause, Gerd
Formato: Artigo
Idioma:Inglês
Publicado em: Portland Press Ltd. 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3561627/
https://ncbi.nlm.nih.gov/pubmed/23356285
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BST20120319
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