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Development of Benzophenone-Alkyne Bifunctional Sigma Receptor Ligands

Sigma (σ) receptors represent unique non-opioid binding sites that are associated with a broad range of disease states. Sigma-2 receptors provide a promising target for diagnostic imaging and pharmacological interventions to curb tumor progression. Most recently, the progesterone receptor (PGRMC1, 2...

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Autors principals: Guo, Lian-Wang, Hajipour, Abdol R., Karaoglu, Kerim, Mavlyutov, Timur A., Ruoho, Arnold E.
Format: Artigo
Idioma:Inglês
Publicat: 2012
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3517089/
https://ncbi.nlm.nih.gov/pubmed/23001760
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cbic.201200427
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