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A Versatile Synthesis of Substituted Isoquinolines

A new and versatile synthesis of substituted isoquinolines: lithiated o-tolualdehyde tert-butylimines are shown to condense with nitriles to form eneamido anion intermediates that can be trapped in situ with various electrophiles, affording a diverse array of highly substituted isoquinolines, many o...

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Autores principales: Si, Chong, Myers, Andrew G.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2011
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3517056/
https://ncbi.nlm.nih.gov/pubmed/21910199
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201104769
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