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Synthesis of Tetrahydropyridazines by a Metal-carbene Directed Highly Enantioselective Vinylogous N-H Insertion/Lewis Acid Catalyzed Diastereoselective Mannich Addition

A versatile reaction cascade triggered by Rh(II)-catalyzed diazo decomposition followed by a vinylogous N-H insertion/Lewis acid catalyzed Mannich addition that produces highly substituted 1,2,3,6-tetrahydropyridazines in up to 97% ee with high yield and diastereocontrol has been developed.

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Detalhes bibliográficos
Main Authors: Xu, Xinfang, Zavalij, Peter Y., Doyle, Michael P.
Formato: Artigo
Idioma:Inglês
Publicado em: 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3517037/
https://ncbi.nlm.nih.gov/pubmed/22945294
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201203962
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