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β-Arrestins specifically constrain β2-adrenergic receptor signaling and function in airway smooth muscle

Chronic use of inhaled beta-agonists by asthmatics is associated with a loss of bronchoprotective effect and deterioration of asthma control. Beta-agonist-promoted desensitization of airway smooth muscle beta-2-adrenergic receptors, mediated by G protein-coupled receptor kinases and arrestins, is pr...

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Detalhes bibliográficos
Main Authors: Deshpande, Deepak A., Theriot, Barbara S., Penn, Raymond B., Walker, Julia K. L.
Formato: Artigo
Idioma:Inglês
Publicado em: 2008
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3514410/
https://ncbi.nlm.nih.gov/pubmed/18337459
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1096/fj.07-102459
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