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Noninvasive Determination of 2-[(18)F]-Fluoroisonicotinic Acid Hydrazide Pharmacokinetics by Positron Emission Tomography in Mycobacterium tuberculosis-Infected Mice

Tuberculosis (TB) is a global pandemic requiring sustained therapy to facilitate curing and to prevent the emergence of drug resistance. There are few adequate tools to evaluate drug dynamics within infected tissues in vivo. In this report, we evaluated a fluorinated analog of isoniazid (INH), 2-[(1...

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Detalhes bibliográficos
Main Authors: Weinstein, E. A., Liu, L., Ordonez, A. A., Wang, H., Hooker, J. M., Tonge, P. J., Jain, S. K.
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3497161/
https://ncbi.nlm.nih.gov/pubmed/23006755
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01644-12
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