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Inactivation of the Cullin (CUL)-RING E3 ligase by the NEDD8-activating enzyme inhibitor MLN4924 triggers protective autophagy in cancer cells

The multiunit Cullin (CUL)-RING E3 ligase (CRL) controls diverse biological processes by targeting a mass of substrates for ubiquitination and degradation, whereas its dysfunction causes carcinogenesis. Post-translational neddylation of CUL, a process triggered by the NEDD8-activating enzyme E1 subu...

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Autors principals: Luo, Zhongguang, Pan, Yongfu, Jeong, Lak Shin, Liu, Jie, Jia, Lijun
Format: Artigo
Idioma:Inglês
Publicat: Landes Bioscience 2012
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3494597/
https://ncbi.nlm.nih.gov/pubmed/22874562
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4161/auto.21484
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