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Therapeutic modulation of cannabinoid lipid signaling: metabolic profiling of a novel antinociceptive cannabinoid-2 receptor agonist

AIMS: AM-1241, a novel, racemic cannabinoid-2 receptor (CB2) ligand, is the primary experimental agonist used to characterize the role of CB2-mediated lipid signaling in health and disease, including substance abuse disorders. In vivo pharmacological effects have been used as indirect proxies for AM...

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Detalles Bibliográficos
Main Authors: Wood, JodiAnne T., Smith, Dustin M., Janero, David R., Zvonok, Alexander M., Makriyannis, Alexandros
Formato: Artigo
Idioma:Inglês
Publicado: 2012
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3493696/
https://ncbi.nlm.nih.gov/pubmed/22749867
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.lfs.2012.06.019
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