Загрузка...

Contribution of Itraconazole Metabolites to Inhibition of CYP3A4 in vivo

Itraconazole (ITZ) is metabolized in vitro to three inhibitory metabolites: hydroxy-ITZ (OH-ITZ), keto-ITZ, and N-desalkyl-ITZ (ND-ITZ). The goal of this study was to determine the contribution of these metabolites to drug-drug interactions caused by ITZ. Six healthy volunteers received 100 mg ITZ o...

Полное описание

Сохранить в:
Библиографические подробности
Главные авторы: Templeton, Ian, Thummel, Kenneth E, Kharasch, Evan D, Kunze, Kent L, Hoffer, Christine, Nelson, Wendel L, Isoherranen, Nina
Формат: Artigo
Язык:Inglês
Опубликовано: 2007
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3488349/
https://ncbi.nlm.nih.gov/pubmed/17495874
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.clpt.6100230
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!