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Bioactivation of Nevirapine to a Reactive Quinone Methide: Implications for Liver Injury

[Image: see text] Nevirapine (NVP) treatment is associated with a significant incidence of liver injury. We developed an anti-NVP antiserum to determine the presence and pattern of covalent binding of NVP to mouse, rat, and human hepatic tissues. Covalent binding to hepatic microsomes from male C57B...

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Bibliographic Details
Main Authors: Sharma, Amy M., Li, Yan, Novalen, Maria, Hayes, M. Anthony, Uetrecht, Jack
Format: Artigo
Language:Inglês
Published: American Chemical Society 2012
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC3475366/
https://ncbi.nlm.nih.gov/pubmed/22793666
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/tx300172s
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