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Macrophages Sequester Clofazimine in an Intracellular Liquid Crystal-Like Supramolecular Organization

Clofazimine is a poorly-soluble but orally-bioavailable small molecule drug that massively accumulates in macrophages when administered over prolonged periods of time. To determine whether crystal-like drug inclusions (CLDIs) that form in subcellular spaces correspond to pure clofazimine crystals, m...

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Autors principals: Baik, Jason, Rosania, Gus R.
Format: Artigo
Idioma:Inglês
Publicat: Public Library of Science 2012
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3469554/
https://ncbi.nlm.nih.gov/pubmed/23071814
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0047494
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