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Design and Functional Characterization of a Novel, Arrestin-Biased Designer G Protein-Coupled Receptor

Mutational modification of distinct muscarinic receptor subtypes has yielded novel designer G protein-coupled receptors (GPCRs) that are unable to bind acetylcholine (ACh), the endogenous muscarinic receptor ligand, but can be efficiently activated by clozapine-N-oxide (CNO), an otherwise pharmacolo...

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Hlavní autoři: Nakajima, Ken-ichiro, Wess, Jürgen
Médium: Artigo
Jazyk:Inglês
Vydáno: The American Society for Pharmacology and Experimental Therapeutics 2012
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3463219/
https://ncbi.nlm.nih.gov/pubmed/22821234
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.112.080358
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