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The A(2) Adenosine Receptor: Guanine Nucleotide Modulation of Agonist Binding Is Enhanced by Proteolysis

Agonist binding to the A(2) adenosine receptor (A(2)AR) and its regulation by guanine nucleotides was studied using the newly developed radioligand (125)l-2-[4-(2-{2-[(4-ammnophenyl)methylcarbonylamino]ethylaminnocarbonyl}ethyl)phenyl]ethylamino-5′-N-ethylcarboxamidoadenosine ((125)1-PAPA-APEC) and...

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Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Prif Awduron: NANOFF, CHRISTIAN, JACOBSON, KENNETH A., STILES, GARY L.
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 1991
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC3463105/
https://ncbi.nlm.nih.gov/pubmed/1899902
Tagiau: Ychwanegu Tag
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