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A Basis for Reduced Chemical Library Inhibition of Firefly Luciferase Obtained from Directed Evolution

We measured the “druggability” of the ATP-dependent luciferase derived from the firefly Photuris pennsylvanica that was optimized using directed evolution (Ultra-Glo™, Promega). Quantitative high throughput screening (qHTS) was used to determine IC(50)’s of 198,899 samples against a formulation of U...

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Bibliografski detalji
Glavni autori: Auld, Douglas S., Zhang, Ya-Qin, Southall, Noel T., Rai, Ganesha, Landsman, Marc, MacLure, Jennifer, Langevin, Daniel, Thomas, Craig J., Austin, Christopher P., Inglese, James
Format: Artigo
Jezik:Inglês
Izdano: 2009
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3430137/
https://ncbi.nlm.nih.gov/pubmed/19215089
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm8014525
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