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Discovery of novel 2-aryl-4-benzoyl-imidazole (ABI–III) analogues targeting tubulin polymerization as antiproliferative agents

Novel ABI–III compounds were designed and synthesized based on our previously reported ABI-I and ABI–II analogs. ABI–III compounds are highly potent against a panel of melanoma and prostate cancer cell lines, with the best compound having an average IC(50) value of 3.8 nM. They are not substrate of...

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Autores principales: Chen, Jianjun, Ahn, Sunjoo, Wang, Jin, Lu, Yan, Dalton, James T., Miller, Duane D., Li, Wei
Formato: Artigo
Lenguaje:Inglês
Publicado: 2012
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3426659/
https://ncbi.nlm.nih.gov/pubmed/22783954
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm300564b
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