Receptor Activity and Conformational Analysis of 5’-Halogenated Resiniferatoxin Analogues as TRPV1 Ligands

A series of 5’-halogenated resiniferatoxin analogues have been investigated in order to examine the effect of halogenation in the A-region on their binding and the functional pattern of agonism/antagonism for rat TRPV1 heterologously expressed in Chinese hamster ovary cells. Halogenation at the 5-po...

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Bibliographische Detailangaben
Hauptverfasser: Lim, Kwang Su, Kang, Dong Wook, Kim, Yong Soo, Kim, Myeong Seop, Park, Seul-Gi, Choi, Sun, Pearce, Larry V., Blumberg, Peter M., Lee, Jeewoo
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2010
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Article
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3420360/
https://ncbi.nlm.nih.gov/pubmed/21111618
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2010.11.012
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