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Pharmacokinetics of dasatinib for Philadelphia-positive acute lymphocytic leukemia with acquired T315I mutation

BACKGROUND: The BCR-ABL T315I kinase domain mutation is insensitive to dasatinib therapy for Philadelphia-positive acute lymphoid leukemia (Ph + ALL) patients. Resistant T315I clone may be present prior to initiating dasatinib, which could expand under selective pressures during treatment. However,...

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Detalhes bibliográficos
Main Authors: Takahashi, Naoto, Miura, Masatomo, Scott, Stuart A, Niioka, Takenori, Sawada, Kenichi
Formato: Artigo
Idioma:Inglês
Publicado em: BioMed Central 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3409074/
https://ncbi.nlm.nih.gov/pubmed/22587422
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/1756-8722-5-23
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