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Physiologically Based Pharmacokinetic Modeling to Investigate Regional Brain Distribution Kinetics in Rats

One of the major challenges in the development of central nervous system (CNS)-targeted drugs is predicting CNS exposure in human from preclinical data. In this study, we present a methodology to investigate brain disposition in rats using a physiologically based modeling approach aiming at improvin...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Westerhout, Joost, Ploeger, Bart, Smeets, Jean, Danhof, Meindert, de Lange, Elizabeth C. M.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Springer US 2012
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC3385827/
https://ncbi.nlm.nih.gov/pubmed/22588644
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-012-9366-1
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