Llwytho...

Selective and cell-active inhibitors of the USP1/UAF1 deubiquitinase complex reverse cisplatin resistance in non-small cell lung cancer cells

Ubiquitin-specific proteases (USPs) have in recent years emerged as a promising therapeutic target class. We identified selective small-molecule inhibitors against a deubiquitinase complex, the human USP1/UAF1, through quantitative high throughput screening (qHTS) of a collection of bioactive molecu...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Prif Awduron: Chen, Junjun, Dexheimer, Thomas S., Ai, Yongxing, Liang, Qin, Villamil, Mark A., Inglese, James, Maloney, David J, Jadhav, Ajit, Simeonov, Anton, Zhuang, Zhihao
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2011
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC3344384/
https://ncbi.nlm.nih.gov/pubmed/22118673
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2011.08.014
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