Caricamento...

p-Anilinoaniline Enhancement of Dioxin-Induced CYP1A1 Transcription and Aryl Hydrocarbon Receptor Occupancy of CYP1A1 Promoter: Role of the Cell Cycle

The aryl hydrocarbon receptor (AhR) is targeted by ubiquitination for degradation by the proteasome shortly after its activation by 2,3,7,8-tetrachlorodibenzo-p-dioxin (TCDD). In silico screening identified p-anilinoaniline (pAA) as a putative inhibitor of an E2 ligase that partners with an E3 ligas...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Autori principali: Elliott, Althea, Joiakim, Aby, Mathieu, Patricia A., Duniec-Dmuchowski, Zofia, Kocarek, Thomas A., Reiners, John J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2012
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3336796/
https://ncbi.nlm.nih.gov/pubmed/22344700
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.111.042549
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !