Cargando...

Human Pregnane X Receptor Activation and CYP3A4/CYP2B6 Induction by 2,3-Oxidosqualene:Lanosterol Cyclase Inhibition

The effects of [4′-(6-allyl-methyl-amino-hexyloxy)-2′-fluoro-phenyl]-(4-bromophenyl)-methanone fumarate (Ro 48-8071), an inhibitor of 2,3-oxidosqualene:lanosterol cyclase (cyclase), were evaluated on CYP3A4 and CYP2B6 mRNA content in primary cultured human hepatocytes. In seven hepatocyte culture pr...

Descrición completa

Gardado en:
Detalles Bibliográficos
Main Authors: Duniec-Dmuchowski, Zofia, Fang, Hai-Lin, Strom, Stephen C., Ellis, Ewa, Runge-Morris, Melissa, Kocarek, Thomas A.
Formato: Artigo
Idioma:Inglês
Publicado: American Society for Pharmacology and Experimental Therapeutics 2009
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC2680536/
https://ncbi.nlm.nih.gov/pubmed/19158313
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.108.025130
Tags: Engadir etiqueta
Sen Etiquetas, Sexa o primeiro en etiquetar este rexistro!