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3-(N-Arylsulfamoyl)benzamides, Inhibitors of Human Sirtuin Type 2 (SIRT2)

Inhibition of sirtuin 2 (SIRT2) is known to be protective against the toxicity of disease proteins in Parkinson’s and Huntington’s models of neurodegeneration. Previously, we developed SIRT2 inhibitors based on the 3-(N-arylsulfamoyl)benzamide scaffold, including 3-(N-(4-bromophenyl)sulfamoyl)-N-(4-...

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Hlavní autoři: Choi, Soo Hyuk, Quinti, Luisa, Kazantsev, Aleksey G., Silverman, Richard B.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2012
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3326608/
https://ncbi.nlm.nih.gov/pubmed/22446090
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2012.02.089
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