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Small molecule inhibitors of arginyltransferase regulate arginylation-dependent protein degradation, cell motility, and angiogenesis

Posttranslational arginylation mediated by arginyltransferase (ATE1) is an emerging major regulator of embryogenesis and cell physiology. Impairments of ATE1 are implicated in congenital heart defects, obesity, cancer, and neurodegeneration making this enzyme an important therapeutic target, whose p...

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Main Authors: Saha, Sougata, Wang, Junling, Buckley, Brian, Wang, Qingqing, Lilly, Brenda, Chernov, Mikhail, Kashina, Anna
Formato: Artigo
Idioma:Inglês
Publicado: 2012
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3288401/
https://ncbi.nlm.nih.gov/pubmed/22280815
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2012.01.012
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