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Molecular Insights into Human Monoamine Oxidase B Inhibition by the Glitazone Antidiabetes Drugs

[Image: see text] The widely employed antidiabetic drug pioglitazone (Actos) is shown to be a specific and reversible inhibitor of human monoamine oxidase B (MAO B). The crystal structure of the enzyme–inhibitor complex shows that the R-enantiomer is bound with the thiazolidinedione ring near the fl...

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Autores principales: Binda, Claudia, Aldeco, Milagros, Geldenhuys, Werner J., Tortorici, Marcello, Mattevi, Andrea, Edmondson, Dale E.
Formato: Artigo
Lenguaje:Inglês
Publicado: American Chemical Society 2011
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3263826/
https://ncbi.nlm.nih.gov/pubmed/22282722
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml200196p
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