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Identification of Kinase Inhibitors that Target Transcription Initiation by RNA Polymerase II

Our current understanding of eukaryotic transcription has greatly benefited from use of small molecule inhibitors that have delineated multiple regulatory steps in site-specific initiation and elongation of RNA synthesis by multiple forms of RNA polymerase (RNAP). This class of “transcription” drugs...

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Autors principals: Morachis, José M., Huang, Ruo, Emerson, Beverly M.
Format: Artigo
Idioma:Inglês
Publicat: Impact Journals LLC 2011
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3248145/
https://ncbi.nlm.nih.gov/pubmed/21378408
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