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Development of a High-Affinity Inhibitor of the Prostaglandin Transporter

Prostaglandin E(2) (PGE(2)) triggers a vast array of biological signals and physiological events. The prostaglandin transporter (PGT) controls PGE(2) influx and is rate-limiting for PGE(2) metabolism and signaling termination. PGT global knockout mice die on postnatal day 1 from patent ductus arteri...

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Autori principali: Chi, Yuling, Min, Jaeki, Jasmin, Jean-Francois, Lisanti, Michael P., Chang, Young-Tae, Schuster, Victor L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3199986/
https://ncbi.nlm.nih.gov/pubmed/21849625
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.111.181354
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