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Halogen substituents on the aromatic moiety of the tetracaine scaffold improve potency of cyclic nucleotide-gated channel block

A series of new tetracaine derivatives with substituents on the aromatic ring was prepared and evaluated for block of retinal rod cyclic nucleotide-gated (CNG) channels. Aromatic substitutions had little effect starting with the basic tetracaine scaffold, but electron-withdrawing substituents signif...

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Detalhes bibliográficos
Main Authors: Kirk, Sarah R., Andrade, Adriana L., Melich, Kenneth, Jackson, Evan P., Cuellar, Elysia, Karpen, Jeffrey W.
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3190055/
https://ncbi.nlm.nih.gov/pubmed/21944857
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2011.08.092
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