Cargando...

Probing the Architecture of an L-type Calcium Channel with a Charged Phenylalkylamine: EVIDENCE FOR A WIDELY OPEN PORE AND DRUG TRAPPING

Voltage-gated calcium channels are in a closed conformation at rest and open temporarily when the membrane is depolarized. To gain insight into the molecular architecture of Ca(v)1.2, we probed the closed and open conformations with the charged phenylalkylamine (−)devapamil ((−)qD888). To elucidate...

Descripción completa

Guardado en:
Detalles Bibliográficos
Autores principales: Beyl, Stanislav, Timin, Eugen N., Hohaus, Annette, Stary, Anna, Kudrnac, Michaela, Guy, Robert H., Hering, Steffen
Formato: Artigo
Lenguaje:Inglês
Publicado: 2006
Materias:
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3189693/
https://ncbi.nlm.nih.gov/pubmed/17138559
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M609153200
Etiquetas: Agregar Etiqueta
Sin Etiquetas, Sea el primero en etiquetar este registro!