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New Betulinic Acid Derivatives as Potent Proteasome Inhibitors

In this study, 22 new betulinic acid (BA) derivatives were synthesized and tested for their inhibition of the chymotrypsin-like activity of 20S proteasome. From the SAR study, we concluded that the C-3 and C-30 positions are the pharmacophores for increasing the proteasome inhibition effects, and la...

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Autori principali: Qian, Keduo, Kim, Sang-Yong, Hung, Hsin-Yi, Huang, Li, Chen, Chin-Ho, Lee, Kuo-Hsiung
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3171619/
https://ncbi.nlm.nih.gov/pubmed/21856154
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2011.07.072
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