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Agonist Derived Molecular Probes for A(2A) Adenosine Receptors

The adenosine agonist 2-(4-(2-carboxyethyl)phenylethylamino)-5′-N-ethylcarboxamidoadenosine (CGS21680) was recently reported to be selective for the A(2A) adenosine receptor subtype, which mediates its hypotensive action. To investigate structurelactivity relationships at a distal site, CGS21680 was...

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Dades bibliogràfiques
Autors principals: Jacobson, Kenneth A., Pannell, Lewis K., Ji, Xiao-duo, Jarvis, Michael F., Williams, Michael, Hutchison, Alan J., Barrington, William W., Stiles, Gary L.
Format: Artigo
Idioma:Inglês
Publicat: 1989
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3157953/
https://ncbi.nlm.nih.gov/pubmed/2561548
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jmr.300020406
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