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In Vivo PET-imaging of Histone Deacetylases by 18F-Suberoylanilide Hydroxamic Acid ((18)F-SAHA)()

Histone deacetylases (HDACs) are a group of enzymes that modulate gene expression and cell state by deacetylation of both histone and non-histone proteins. A variety of HDAC inhibitors (HDACi) have already undergone clinical testing in cancer. Real-time in vivo imaging of HDACs and their inhibition...

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Autores principales: Hendricks, J. Adam, Keliher, Edmund J., Marinelli, Brett, Reiner, Thomas, Weissleder, Ralph, Mazitschek, Ralph
Formato: Artigo
Lenguaje:Inglês
Publicado: 2011
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3150598/
https://ncbi.nlm.nih.gov/pubmed/21721525
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm200620f
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