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Design of novel melanocortin receptor ligands: multiple receptors, complex pharmacology, the challenge

The major pharmacophore for the melanocortin 1,3,4 and 5 receptors is the sequence -His-Phe-Arg-Trp-. There is a need for potent, biologically stable, receptor selective ligands, both agonists and antagonists, for these receptors. In this report we briefly examine the structural and biophysical appr...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Hruby, Victor J., Cai, Minying, Cain, James, Nyberg, Joel, Trivedi, Dev
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2011
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3138524/
https://ncbi.nlm.nih.gov/pubmed/21208601
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejphar.2010.10.109
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