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Single enantiomer synthesis of α-(trifluoromethyl)-β-lactam

The first synthesis of α-(trifluoromethyl)-β-lactam ((S)-1) is reported. The route starts from α-(trifluoromethyl)acrylic acid (2). Conjugate addition of α-(p-methoxyphenyl)ethylamine ((S)-3b), generated an addition adduct 4b which was cyclised to β-lactam 5b. Separation of the diastereoisomers by c...

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Detalhes bibliográficos
Main Authors: Jurčík, Václav, Slawin, Alexandra M Z, O'Hagan, David
Formato: Artigo
Idioma:Inglês
Publicado em: Beilstein-Institut 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3135179/
https://ncbi.nlm.nih.gov/pubmed/21804871
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.7.86
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