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Ligand binding domain mutations of glucocorticoid receptor selectively modify effects with, but not binding of, cofactors

We previously reported that several point mutations in the ligand binding domain (LBD) of glucocorticoid receptors (GRs) marginally affect the binding affinity of the synthetic glucocorticoids dexamethasone (Dex) and deacylcortivazol (DAC). However, these mutations dramatically alter the efficacy (A...

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Detalhes bibliográficos
Main Authors: Lee, Geun-Shik, Simons, S. Stoney
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3123670/
https://ncbi.nlm.nih.gov/pubmed/21142156
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi101792d
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