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Dual-Functional, Receptor-Targeted Fluorogenic Probe for In Vivo Imaging of Extracellular Protease Expressions

Herein we report a new type of in vivo fluorogenic probe that enables simultaneous and active targeting of overexpressed receptors, α(v)β(3) integrins, and extracellular proteases, matrix metalloproteinases (MMPs), in the tumor regions. This c(RGDyK)-conjugated MMP fluorogenic probe efficiently targ...

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Dettagli Bibliografici
Autori principali: Zhu, Lei, Xie, Jin, Swierczewska, Magdalena, Zhang, Fan, Lin, Xin, Fang, Xuexun, Niu, Gang, Lee, Seulki, Chen, Xiaoyuan
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3118575/
https://ncbi.nlm.nih.gov/pubmed/21574650
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bc200005w
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