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Contributions of the D-Ring to the Activity of Etoposide Against Human Topoisomerase IIα: Potential Interactions with DNA in the Ternary Enzyme-Drug-DNA Complex

Etoposide is a widely prescribed anticancer drug that stabilizes covalent topoisomerase II-cleaved DNA complexes. The drug contains a polycyclic ring system (rings A–D), a glycosidic moiety at C4, and a pendant ring (E–ring) at C1. Interactions between human topoisomerase IIα and etoposide in the bi...

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Bibliografski detalji
Glavni autori: Pitts, Steven L., Jablonksy, Michael J., Duca, Maria, Dauzonne, Daniel, Monneret, Claude, Arimondo, Paola B., Anklin, Clemens, Graves, David E., Osheroff, Neil
Format: Artigo
Jezik:Inglês
Izdano: 2011
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3109987/
https://ncbi.nlm.nih.gov/pubmed/21548574
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi200531q
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