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Utilization of Nitrophenylphosphates and Oxime-Based Ligation for the Development of Nanomolar Affinity Inhibitors of the Yersinia Pestis Outer Protein H (YopH) Phosphatase, ,

Our current study reports the first K(M) optimization of a library of nitrophenylphosphate-containing substrates for generating an inhibitor lead against the Yersinia pestis outer protein phosphatase (YopH). A high activity substrate identified by this method (K(M) = 80 μM was converted from a subst...

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Detalhes bibliográficos
Main Authors: Bahta, Medhanit, Lountos, George T., Dyas, Beverly, Kim, Sung-Eun, Ulrich, Robert G., Waugh, David S., Burke, Terrence R.
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3085962/
https://ncbi.nlm.nih.gov/pubmed/21443195
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm200022g
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