Chargement en cours...

Asymmetric Synthesis of 1,2,9,9a-Tetrahydrocyclopropa[c]benzo[e]indol-4-one (CBI)

A short, asymmetric synthesis of the 1,2,9,9a-tetrahydrocyclopropa[c]benzo[e]indol-4-one (CBI) analogue of the CC-1065 and duocarmycin DNA alkylation subunits is described. Treatment of iodo-epoxide 5, prepared by late-stage alkylation of 4 with (S)-glycidal-3-nosylate, with EtMgBr at room temperatu...

Description complète

Enregistré dans:
Détails bibliographiques
Auteurs principaux: Lajiness, James P., Boger, Dale L.
Format: Artigo
Langue:Inglês
Publié: 2010
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3079324/
https://ncbi.nlm.nih.gov/pubmed/21192653
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jo102136w
Tags: Ajouter un tag
Pas de tags, Soyez le premier à ajouter un tag!