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Structure-activity relationship study of 2,4-diaminothiazoles as cdk5/p25 kinase inhibitors

Cdk5/p25 has emerged as a principle therapeutic target for numerous acute and chronic neurodegenerative diseases, including Alzheimer’s disease. A structure-activity relationship study of 2,4-diaminothiazole inhibitors revealed that increased Cdk5/p25 inhibitory activity could be accomplished by inc...

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Hlavní autoři: Laha, Joydev K., Zhang, Xuemei, Qiao, Lixin, Liu, Min, Chatterjee, Snigdha, Robinson, Shaughnessy, Kosik, Kenneth S., Cuny, Gregory D.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2011
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3062192/
https://ncbi.nlm.nih.gov/pubmed/21353545
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2011.01.140
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