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Phenolic Bis-Styrylbenzenes as β-Amyloid Binding Ligands and Free Radical Scavengers
Starting from bisphenolic bis-styrylbenzene DF-9 (4), β-amyloid (Aβ) binding affinity and specificity for phenolic bis-styrylbenzenes, mono-styrylbenzenes and alkyne controls were determined by fluorescence titration with β-amyloid peptide Aβ(1-40) and a fluorescence assay using APP/PS1 transgenic m...
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| Autores principales: | , , , , |
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| Formato: | Artigo |
| Lenguaje: | Inglês |
| Publicado: |
2010
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| Materias: | |
| Acceso en línea: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3057505/ https://ncbi.nlm.nih.gov/pubmed/21038854 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm1006929 |
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