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Participation of CYP2C8 and CYP3A4 in the N-demethylation of imatinib in human hepatic microsomes

BACKGROUND AND PURPOSE: Imatinib is a clinically important inhibitor of tyrosine kinases that are dysregulated in chronic myelogenous leukaemia and gastrointestinal stromal tumours. Inter-individual variation in imatinib pharmacokinetics is extensive, and influences drug safety and efficacy. Hepatic...

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Détails bibliographiques
Auteurs principaux: Nebot, Noelia, Crettol, Severine, d'Esposito, Fabrizio, Tattam, Bruce, Hibbs, David E, Murray, Michael
Format: Artigo
Langue:Inglês
Publié: Blackwell Publishing Ltd 2010
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Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2998687/
https://ncbi.nlm.nih.gov/pubmed/20977456
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1476-5381.2010.00946.x
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