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Quantitative Structure Activity Relationship for Inhibition of Human Organic Cation/Carnitine Transporter (OCTN2)

Organic cation/carnitine transporter (OCTN2; SLC22A5) is an important transporter for L-carnitine homeostasis, but can be inhibited by drugs, which may cause L-carnitine deficiency and possibly other OCTN2-mediated drug-drug interactions. One objective was to develop a quantitative structure–activit...

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Main Authors: Diao, Lei, Ekins, Sean, Polli, James E.
Formato: Artigo
Idioma:Inglês
Publicado: 2010
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC2997942/
https://ncbi.nlm.nih.gov/pubmed/20831193
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/mp100226q
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