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Specificity of a Prodrug-Activating Enzyme hVACVase: the Leaving Group Effect

Human valacyclovirase (hVACVase) is a prodrug-activating enzyme for amino acid prodrugs including the antiviral drugs valacyclovir and valganciclovir. In hVACVase-catalyzed reactions, the leaving group of the substrate corresponds to the drug moiety of the prodrug, making the leaving group effect es...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Sun, Jing, Dahan, Arik, Walls, Zachary F., Lai, Longsheng, Lee, Kyung-Dall, Amidon, Gordon L.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2010
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC2997884/
https://ncbi.nlm.nih.gov/pubmed/21028903
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/mp100300k
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