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Novel alpha3beta4 nicotinic acetylcholine receptor-selective ligands. Discovery, structure-activity studies and pharmacological evaluation

Antagonist activity at the alpha3beta4 nicotinic acetylcholine receptor (nAChR) is thought to contribute to the anti-addictive properties of several compounds. However, truly selective ligands for the α3β4 nAChR have not been available. We report the discovery and SAR of a novel class of compounds t...

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Библиографические подробности
Главные авторы: Zaveri, Nurulain, Jiang, Faming, Olsen, Cris, Polgar, Willma, Toll, Lawrence
Формат: Artigo
Язык:Inglês
Опубликовано: 2010
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC2997436/
https://ncbi.nlm.nih.gov/pubmed/20979364
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm1006148
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