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Design and Optimization of Mefloquine Hydrochloride Microparticles for Bitter Taste Masking

The objective of the present investigation was to reduce the bitterness with improved dissolution, in acidic medium (pH 1.2), of mefloquine hydrochloride (MFL). Microparticles were prepared by coacervation method using Eudragit E (EE) as polymer and sodium hydroxide as precipitant. A 3(2) full facto...

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Autori principali: Shah, Punit P., Mashru, Rajashree C., Rane, Yogesh M., Thakkar, Arti
Natura: Artigo
Lingua:Inglês
Pubblicazione: Springer US 2008
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2976944/
https://ncbi.nlm.nih.gov/pubmed/18431670
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12249-008-9052-x
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