Carregant...

Overlapping Binding Sites of Structurally Different Antiarrhythmics Flecainide and Propafenone in the Subunit Interface of Potassium Channel Kv2.1

Kv2.1 channels, which are expressed in brain, heart, pancreas, and other organs and tissues, are important targets for drug design. Flecainide and propafenone are known to block Kv2.1 channels more potently than other Kv channels. Here, we sought to explore structural determinants of this selectivit...

Descripció completa

Guardat en:
Dades bibliogràfiques
Autors principals: Madeja, Michael, Steffen, Wibke, Mesic, Ivana, Garic, Bojan, Zhorov, Boris S.
Format: Artigo
Idioma:Inglês
Publicat: American Society for Biochemistry and Molecular Biology 2010
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2962489/
https://ncbi.nlm.nih.gov/pubmed/20709754
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M110.159897
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!