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Efficient Hypoxic Activation of the Anticancer Agent AQ4N by CYP2S1 and CYP2W1

AQ4N [1,4-bis{[2-(dimethylamino-N-oxide)ethyl]amino}-5,8-dihydroxyanthracene-9,10-dione], a prodrug with two dimethylamino N-oxide groups, is converted to the topoisomerase II inhibitor AQ4 [1,4-bis{[2-(dimethylamino)ethyl]amino}-5,8-dihydroxy-anthracene-9,10-dione] by reduction of the N-oxides to d...

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Detalhes bibliográficos
Main Authors: Nishida, Clinton R., Lee, Melody, de Montellano, Paul R. Ortiz
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2939484/
https://ncbi.nlm.nih.gov/pubmed/20566689
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.110.065045
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