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The transcription inhibitor lipiarmycin blocks DNA fitting into the RNA polymerase catalytic site

Worldwide spreading of drug-resistant pathogens makes mechanistic understanding of antibiotic action an urgent task. The macrocyclic antibiotic lipiarmycin (Lpm), which is under development for clinical use, inhibits bacterial RNA polymerase (RNAP) by an unknown mechanism. Using genetic and biochemi...

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Autori principali: Tupin, Audrey, Gualtieri, Maxime, Leonetti, Jean-Paul, Brodolin, Konstantin
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 2010
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2928680/
https://ncbi.nlm.nih.gov/pubmed/20562828
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/emboj.2010.135
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